+ | 1 | 4BZD | Cyclin dependent kinase 2 CDK2 | ATP domain | 8.61 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 1.83 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 4 |
---|
|
+ | 2 | 1E9H | Cyclin dependent kinase 2 CDK2 | ATP domain | 8.59 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 2.5 Å |
---|
Reference Affinity: | IC50=35nM |
---|
Interaction Features: | 9 |
---|
|
+ | 3 | 1PF8 | Cyclin dependent kinase 2 CDK2 | ATP domain | 8.56 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 2.51 Å |
---|
Reference Affinity: | Ki=0.031uM |
---|
Interaction Features: | 6 |
---|
|
+ | 4 | 4GII | Non-receptor tyrosine-protein kinase TYK2 | ATP domain | 8.43 |
---|
Additional Details |
---|
Target Short Name: | TYK2 |
---|
Cystal Resolution: | 2.31 Å |
---|
Reference Affinity: | Ki=1.8nM |
---|
Interaction Features: | 5 |
---|
|
+ | 5 | 4ZS0 | Aurora A kinase AurA | ATP domain | 8.43 |
---|
Additional Details |
---|
Target Short Name: | AurA |
---|
Cystal Resolution: | 3 Å |
---|
Reference Affinity: | IC50=2.3uM |
---|
Interaction Features: | 5 |
---|
|
+ | 6 | 3LXL | Tyrosine-protein kinase JAK3 | ATP domain | 8.40 |
---|
Additional Details |
---|
Target Short Name: | JAK3 |
---|
Cystal Resolution: | 1.74 Å |
---|
Reference Affinity: | IC50=5nM |
---|
Interaction Features: | 4 |
---|
|
+ | 7 | 6G33 | Dual specificity protein kinase clk1 | ATP domain | 8.38 |
---|
Additional Details |
---|
Target Short Name: | CLK1 |
---|
Cystal Resolution: | 2.05 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 3 |
---|
|
+ | 8 | 2XYN | Tyrosine-protein kinase ABL2 | ATP domain | 8.36 |
---|
Additional Details |
---|
Target Short Name: | ABL2 |
---|
Cystal Resolution: | 2.81 Å |
---|
Reference Affinity: | Kd=4nM |
---|
Interaction Features: | 5 |
---|
|
+ | 9 | 4YTI | Tyrosine-protein kinase JAK2 | ATP domain | 8.36 |
---|
Additional Details |
---|
Target Short Name: | JAK2 |
---|
Cystal Resolution: | 2.52 Å |
---|
Reference Affinity: | Ki=13nM |
---|
Interaction Features: | 4 |
---|
|
+ | 10 | 1X8B | Wee1-like protein kinase WEE1 | ATP domain | 8.34 |
---|
Additional Details |
---|
Target Short Name: | WEE1 |
---|
Cystal Resolution: | 1.81 Å |
---|
Reference Affinity: | IC50=97nM |
---|
Interaction Features: | 8 |
---|
|
+ | 11 | 2XJ2 | Serine/threonine-protein kinase PIM1 | ATP domain | 8.31 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 2.2 Å |
---|
Reference Affinity: | Kd=66nM |
---|
Interaction Features: | 7 |
---|
|
+ | 12 | 3BGZ | Serine/threonine-protein kinase PIM1 | ATP domain | 8.31 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 2.4 Å |
---|
Reference Affinity: | Ki=0.55uM |
---|
Interaction Features: | 7 |
---|
|
+ | 13 | 2WMQ | Serine/threonine-Transferase CHK1 | ATP domain | 8.27 |
---|
Additional Details |
---|
Target Short Name: | CHK1 |
---|
Cystal Resolution: | 2.48 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 3 |
---|
|
+ | 14 | 5AAF | Aurora A kinase AurA | ATP domain | 8.27 |
---|
Additional Details |
---|
Target Short Name: | AurA |
---|
Cystal Resolution: | 2.78 Å |
---|
Reference Affinity: | IC50=0.036uM |
---|
Interaction Features: | 4 |
---|
|
+ | 15 | 5OQ8 | Serine/threonine-Transferase CHK1 | ATP domain | 8.27 |
---|
Additional Details |
---|
Target Short Name: | CHK1 |
---|
Cystal Resolution: | 2 Å |
---|
Reference Affinity: | Ki=1.41uM |
---|
Interaction Features: | 3 |
---|
|
+ | 16 | 6AAK | Tyrosine-protein kinase jak3 | ATP domain | 8.27 |
---|
Additional Details |
---|
Target Short Name: | JAK3 |
---|
Cystal Resolution: | 2.67 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 3 |
---|
|
+ | 17 | 3E63 | Tyrosine-protein kinase JAK2 | ATP domain | 8.27 |
---|
Additional Details |
---|
Target Short Name: | JAK2 |
---|
Cystal Resolution: | 1.9 Å |
---|
Reference Affinity: | IC50=1.6uM |
---|
Interaction Features: | 4 |
---|
|
+ | 18 | 4BBF | Tyrosine-protein kinase JAK2 | ATP domain | 8.25 |
---|
Additional Details |
---|
Target Short Name: | JAK2 |
---|
Cystal Resolution: | 2 Å |
---|
Reference Affinity: | IC50=2.2nM |
---|
Interaction Features: | 5 |
---|
|
+ | 19 | 3E64 | Tyrosine-protein kinase JAK2 | ATP domain | 8.22 |
---|
Additional Details |
---|
Target Short Name: | JAK2 |
---|
Cystal Resolution: | 1.8 Å |
---|
Reference Affinity: | Kd=0.078uM |
---|
Interaction Features: | 5 |
---|
|
+ | 20 | 5OPV | Serine/threonine-Transferase CHK1 | ATP domain | 8.22 |
---|
Additional Details |
---|
Target Short Name: | CHK1 |
---|
Cystal Resolution: | 1.9 Å |
---|
Reference Affinity: | IC50=8nM |
---|
Interaction Features: | 4 |
---|
|
+ | 21 | 3E62 | Tyrosine-protein kinase JAK2 | ATP domain | 8.22 |
---|
Additional Details |
---|
Target Short Name: | JAK2 |
---|
Cystal Resolution: | 1.92 Å |
---|
Reference Affinity: | IC50=40.9uM |
---|
Interaction Features: | 4 |
---|
|
+ | 22 | 3ORN | Dual specificity mitogen-activated protein kinase kinase 1 MAP2K1 | ATP domain | 8.22 |
---|
Additional Details |
---|
Target Short Name: | MAP2K1 |
---|
Cystal Resolution: | 2.8 Å |
---|
Reference Affinity: | Kd=0.24nM |
---|
Interaction Features: | 7 |
---|
|
+ | 23 | 2BR1 | Serine/threonine-Transferase CHK1 | ATP domain | 8.22 |
---|
Additional Details |
---|
Target Short Name: | CHK1 |
---|
Cystal Resolution: | 2 Å |
---|
Reference Affinity: | Ki=7.2uM |
---|
Interaction Features: | 3 |
---|
|
+ | 24 | 2Z2W | Wee1-like protein kinase WEE1 | ATP domain | 8.20 |
---|
Additional Details |
---|
Target Short Name: | WEE1 |
---|
Cystal Resolution: | 2.22 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 8 |
---|
|
+ | 25 | 4I4F | Focal adhesion kinase 1 FAK1 | ATP domain | 8.20 |
---|
Additional Details |
---|
Target Short Name: | FAK1 |
---|
Cystal Resolution: | 1.75 Å |
---|
Reference Affinity: | IC50=0.64uM |
---|
Interaction Features: | 7 |
---|
|
+ | 26 | 4XV9 | Serine/threonine-protein kinase BRAF | ATP domain/Hydrophobic pocket | 8.20 |
---|
Additional Details |
---|
Target Short Name: | BRAF |
---|
Cystal Resolution: | 2 Å |
---|
Reference Affinity: | IC50=0.19uM |
---|
Interaction Features: | 9 |
---|
|
+ | 27 | 3F2A | Serine/threonine-protein kinase PIM1 | ATP domain | 8.20 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 1.9 Å |
---|
Reference Affinity: | IC50=57nM |
---|
Interaction Features: | 7 |
---|
|
+ | 28 | 2BRO | Serine/threonine-Transferase CHK1 | ATP domain | 8.20 |
---|
Additional Details |
---|
Target Short Name: | CHK1 |
---|
Cystal Resolution: | 2.2 Å |
---|
Reference Affinity: | IC50=1.4uM |
---|
Interaction Features: | 4 |
---|
|
+ | 29 | 2XIZ | Serine/threonine-protein kinase PIM1 | ATP domain | 8.18 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 2.21 Å |
---|
Reference Affinity: | IC50=130uM |
---|
Interaction Features: | 4 |
---|
|
+ | 30 | 3VBX | Serine/threonine-protein kinase PIM1 | ATP domain | 8.18 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 2.03 Å |
---|
Reference Affinity: | IC50=17uM |
---|
Interaction Features: | 4 |
---|
|
+ | 31 | 2VTQ | Cyclin dependent kinase 2 CDK2 | ATP domain | 8.18 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 1.9 Å |
---|
Reference Affinity: | IC50=140nM |
---|
Interaction Features: | 4 |
---|
|
+ | 32 | 4USF | STE20-like serine/threonine-protein kinase | ATP domain | 8.18 |
---|
Additional Details |
---|
Target Short Name: | SLK |
---|
Cystal Resolution: | 1.75 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 6 |
---|
|
+ | 33 | 3PIY | Tyrosine-protein kinase BTK | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | BTK |
---|
Cystal Resolution: | 2.55 Å |
---|
Reference Affinity: | IC50=0.29uM |
---|
Interaction Features: | 6 |
---|
|
+ | 34 | 5CT0 | Casein kinase II subunit alpha CK2A1 | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | CK2A1 |
---|
Cystal Resolution: | 2.01 Å |
---|
Reference Affinity: | Kd=270uM |
---|
Interaction Features: | 6 |
---|
|
+ | 35 | 3HUC | Mitogen-activated protein kinase 14 MAPK14 | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | MAPK14 |
---|
Cystal Resolution: | 1.8 Å |
---|
Reference Affinity: | Kd=1030nM |
---|
Interaction Features: | 7 |
---|
|
+ | 36 | 2OW3 | Glycogen synthase kinase-3 beta GSK3B | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | GSK3B |
---|
Cystal Resolution: | 2.8 Å |
---|
Reference Affinity: | IC50=3nM |
---|
Interaction Features: | 6 |
---|
|
+ | 37 | 5P9L | Tyrosine-protein kinase BTK | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | BTK |
---|
Cystal Resolution: | 1.25 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 5 |
---|
|
+ | 38 | 5QIN | TGF-beta receptor type-2 TGFBR2 | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | TGFBR2 |
---|
Cystal Resolution: | 1.57 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 8 |
---|
|
+ | 39 | 3NUY | Phosphoinositide-dependent kinase-1 PDK1 | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | PDPK1 |
---|
Cystal Resolution: | 2.1 Å |
---|
Reference Affinity: | IC50=345uM |
---|
Interaction Features: | 3 |
---|
|
+ | 40 | 2OIC | Interleukin-1 receptor-associated kinase 4 IRAK4 | ATP domain | 8.15 |
---|
Additional Details |
---|
Target Short Name: | IRAK4 |
---|
Cystal Resolution: | 2.4 Å |
---|
Reference Affinity: | IC50=4nM |
---|
Interaction Features: | 7 |
---|
|
+ | 41 | 2XJ0 | Serine/threonine-protein kinase PIM1 | ATP domain | 8.13 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 3.1 Å |
---|
Reference Affinity: | IC50=1500uM |
---|
Interaction Features: | 4 |
---|
|
+ | 42 | 5UT5 | Tyrosine-protein kinase JAK2 | ATP domain | 8.13 |
---|
Additional Details |
---|
Target Short Name: | JAK2 |
---|
Cystal Resolution: | 1.9 Å |
---|
Reference Affinity: | Kd=50uM |
---|
Interaction Features: | 5 |
---|
|
+ | 43 | 3CR0 | Wee1-like protein kinase WEE1 | ATP domain | 8.13 |
---|
Additional Details |
---|
Target Short Name: | WEE1 |
---|
Cystal Resolution: | 2.3 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 8 |
---|
|
+ | 44 | 5L2S | Cyclin-dependent kinase 6 CDK6 | ATP domain | 8.13 |
---|
Additional Details |
---|
Target Short Name: | CDK6 |
---|
Cystal Resolution: | 2.27 Å |
---|
Reference Affinity: | Kd=83nM |
---|
Interaction Features: | 10 |
---|
|
+ | 45 | 5CI7 | Serine/threonine-protein kinase ULK1 | ATP domain | 8.11 |
---|
Additional Details |
---|
Target Short Name: | ULK1 |
---|
Cystal Resolution: | 1.74 Å |
---|
Reference Affinity: | IC50=120nM |
---|
Interaction Features: | 3 |
---|
|
+ | 46 | 3R01 | Serine/threonine-protein kinase PIM1 | ATP domain | 8.11 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 2.6 Å |
---|
Reference Affinity: | IC50=5.8uM |
---|
Interaction Features: | 5 |
---|
|
+ | 47 | 4JAJ | Aurora A kinase AurA | ATP domain | 8.11 |
---|
Additional Details |
---|
Target Short Name: | AurA |
---|
Cystal Resolution: | 2.7 Å |
---|
Reference Affinity: | IC50=5.54uM |
---|
Interaction Features: | 3 |
---|
|
+ | 48 | 4RJ7 | Epidermal growth factor receptor EGFR | ATP domain | 8.11 |
---|
Additional Details |
---|
Target Short Name: | EGFR |
---|
Cystal Resolution: | 2.55 Å |
---|
Reference Affinity: | Ki=22nM |
---|
Interaction Features: | 5 |
---|
|
+ | 49 | 4HVB | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | ATP domain | 8.11 |
---|
Additional Details |
---|
Target Short Name: | PIK3CG |
---|
Cystal Resolution: | 2.35 Å |
---|
Reference Affinity: | Ki=0.111nM |
---|
Interaction Features: | 8 |
---|
|
+ | 50 | 5DXH | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform | ATP domain | 8.09 |
---|
Additional Details |
---|
Target Short Name: | PIK3CA |
---|
Cystal Resolution: | 3 Å |
---|
Reference Affinity: | Ki=0.2nM |
---|
Interaction Features: | 6 |
---|
|
+ | 51 | 1Y6B | Vascular endothelial growth factor receptor 2 VEGFR2 | ATP domain | 8.09 |
---|
Additional Details |
---|
Target Short Name: | VEGFR2 |
---|
Cystal Resolution: | 2.1 Å |
---|
Reference Affinity: | IC50=38nM |
---|
Interaction Features: | 7 |
---|
|
+ | 52 | 4QPS | Tyrosine-protein kinase JAK3 | ATP domain | 8.09 |
---|
Additional Details |
---|
Target Short Name: | JAK3 |
---|
Cystal Resolution: | 1.8 Å |
---|
Reference Affinity: | IC50=0.30uM |
---|
Interaction Features: | 3 |
---|
|
+ | 53 | 4Y72 | Cyclin-dependent kinase 1 CDK1 | ATP domain | 8.07 |
---|
Additional Details |
---|
Target Short Name: | CDK1 |
---|
Cystal Resolution: | 2.3 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 5 |
---|
|
+ | 54 | 4F65 | Fibroblast growth factor receptor 1 FGFR1 | ATP domain | 8.06 |
---|
Additional Details |
---|
Target Short Name: | FGFR1 |
---|
Cystal Resolution: | 2.26 Å |
---|
Reference Affinity: | IC50=2.5nM |
---|
Interaction Features: | 6 |
---|
|
+ | 55 | 5N4V | Serine/threonine-protein kinase PIM1 | ATP domain | 8.06 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 1.85 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 6 |
---|
|
+ | 56 | 6CCF | Calcium/calmodulin-dependent protein kinase kinase 1 CAMK1 | ATP domain | 8.06 |
---|
Additional Details |
---|
Target Short Name: | CAMK1 |
---|
Cystal Resolution: | 2.10 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 6 |
---|
|
+ | 57 | 4BB4 | Ephrin type-B receptor 4 EPHB4 | ATP domain | 8.06 |
---|
Additional Details |
---|
Target Short Name: | EPHB4 |
---|
Cystal Resolution: | 1.65 Å |
---|
Reference Affinity: | IC50=190nM |
---|
Interaction Features: | 7 |
---|
|
+ | 58 | 5QIM | TGF-beta receptor type I TGFBR1 | ATP domain | 8.04 |
---|
Additional Details |
---|
Target Short Name: | TGFBR1 |
---|
Cystal Resolution: | 1.75 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 6 |
---|
|
+ | 59 | 3W32 | Epidermal growth factor receptor EGFR | ATP domain | 8.04 |
---|
Additional Details |
---|
Target Short Name: | EGFR |
---|
Cystal Resolution: | 1.8 Å |
---|
Reference Affinity: | IC50=75nM |
---|
Interaction Features: | 8 |
---|
|
+ | 60 | 5A4Q | Dual specificity tyrosine-phosphorylation-regulated kinase 1A DYRK1A | ATP domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | DYRK1A |
---|
Cystal Resolution: | 2.37 Å |
---|
Reference Affinity: | IC50=2.9uM |
---|
Interaction Features: | 3 |
---|
|
+ | 61 | 4PS5 | Bromodomain-containing protein 4 | BRD domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | BRD4 |
---|
Cystal Resolution: | 1.40 Å |
---|
Reference Affinity: | IC50=0.29uM |
---|
Interaction Features: | 6 |
---|
|
+ | 62 | 3LFS | Cyclin dependent kinase 2 CDK2 | ATP domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 2.4 Å |
---|
Reference Affinity: | IC50=2500nM |
---|
Interaction Features: | 3 |
---|
|
+ | 63 | 3DOG | Cyclin dependent kinase 2 CDK2 | ATP domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 2.7 Å |
---|
Reference Affinity: | IC50=0.04uM |
---|
Interaction Features: | 4 |
---|
|
+ | 64 | 4L3J | Ribosomal protein S6 kinase beta-1 PRS6KB1 | ATP domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | RPS6KB1 |
---|
Cystal Resolution: | 2.1 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 3 |
---|
|
+ | 65 | 5F60 | Bromodomain-containing protein 4 | BRD domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | BRD4 |
---|
Cystal Resolution: | 1.35 Å |
---|
Reference Affinity: | Kd=43nM |
---|
Interaction Features: | 7 |
---|
|
+ | 66 | 5F62 | Bromodomain-containing protein 4 | BRD domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | BRD4 |
---|
Cystal Resolution: | 1.35 Å |
---|
Reference Affinity: | Kd=6.8nM |
---|
Interaction Features: | 7 |
---|
|
+ | 67 | 5F63 | Bromodomain-containing protein 4 | BRD domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | BRD4 |
---|
Cystal Resolution: | 1.45 Å |
---|
Reference Affinity: | Kd=12nM |
---|
Interaction Features: | 7 |
---|
|
+ | 68 | 5FP6 | Cyclin dependent kinase 2 CDK2 | ATP domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 1.85 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 8 |
---|
|
+ | 69 | 5J9L | Mitogen-activated protein kinase kinase kinase 7, TGF-beta-activated kinase 1 and MAP3K7-binding proNoin 1 | ATP domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | TAB1 |
---|
Cystal Resolution: | 2.751IC50=34nM Å |
---|
Reference Affinity: | IC50=34nM |
---|
Interaction Features: | 5 |
---|
|
+ | 70 | 5K0X | Tyrosine-protein kinase Mer MERTK | ATP domain | 8.02 |
---|
Additional Details |
---|
Target Short Name: | MERTK |
---|
Cystal Resolution: | 2.231IC50=4.4nM Å |
---|
Reference Affinity: | IC50=4.4nM |
---|
Interaction Features: | 5 |
---|
|
+ | 71 | 5O3F | Bromodomain-containing protein 2 | BRD domain | 8.00 |
---|
Additional Details |
---|
Target Short Name: | BRD2 |
---|
Cystal Resolution: | 1.75 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 5 |
---|
|
+ | 72 | 3R00 | Serine/threonine-protein kinase PIM1 | ATP domain | 8.00 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 2.1 Å |
---|
Reference Affinity: | IC50=8.5uM |
---|
Interaction Features: | 4 |
---|
|
+ | 73 | 2X7G | UNCHARACTERIZED PROTEIN SRPK2 | ATP domain | 8.00 |
---|
Additional Details |
---|
Target Short Name: | SRPK2 |
---|
Cystal Resolution: | 2.5 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 3 |
---|
|
+ | 74 | 4ARK | Dual specificity mitogen-activated protein kinase kinase 1 MAP2K1 | Hydrophobic pocket | 8.00 |
---|
Additional Details |
---|
Target Short Name: | MAP2K1 |
---|
Cystal Resolution: | 2.6 Å |
---|
Reference Affinity: | IC50=63nM |
---|
Interaction Features: | 7 |
---|
|
+ | 75 | 5O12 | Serine/threonine-protein kinase PIM1 | ATP domain | 8.00 |
---|
Additional Details |
---|
Target Short Name: | PIM1 |
---|
Cystal Resolution: | 2.4 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 5 |
---|
|
+ | 76 | 6HM6 | Spleen tyrosine kinase | ATP domain | 8.00 |
---|
Additional Details |
---|
Target Short Name: | SYK |
---|
Cystal Resolution: | 2.10 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 4 |
---|
|
+ | 77 | 5DW2 | Bromodomain-containing protein 4 | BRD domain | 7.97 |
---|
Additional Details |
---|
Target Short Name: | BRD4 |
---|
Cystal Resolution: | 1.12 Å |
---|
Reference Affinity: | Kd=1.44uM |
---|
Interaction Features: | 4 |
---|
|
+ | 78 | 3QGY | Tyrosine-protein kinase ITK/TSK | ATP domain | 7.97 |
---|
Additional Details |
---|
Target Short Name: | ITK |
---|
Cystal Resolution: | 2.1 Å |
---|
Reference Affinity: | Ki=16nM |
---|
Interaction Features: | 6 |
---|
|
+ | 79 | 6BRJ | Epithelial discoidin domain-containing receptor 1 DDR1 | ATP domain | 7.97 |
---|
Additional Details |
---|
Target Short Name: | DDR1 |
---|
Cystal Resolution: | 2.231~ Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 3 |
---|
|
+ | 80 | 5N7V | Dual specificity protein kinase TTK | ATP domain | 7.97 |
---|
Additional Details |
---|
Target Short Name: | TTK |
---|
Cystal Resolution: | 2.52 Å |
---|
Reference Affinity: | IC50=1.9nM |
---|
Interaction Features: | 4 |
---|
|
+ | 81 | 3COH | Serine/threonine-Transferase 6 STK6 | ATP domain | 7.97 |
---|
Additional Details |
---|
Target Short Name: | STK6 |
---|
Cystal Resolution: | 2.7 Å |
---|
Reference Affinity: | IC50=4nM |
---|
Interaction Features: | 3 |
---|
|
+ | 82 | 3LQ5 | Cyclin-dependent kinase 9 CDK9 | ATP domain | 7.97 |
---|
Additional Details |
---|
Target Short Name: | CDK9 |
---|
Cystal Resolution: | 3 Å |
---|
Reference Affinity: | IC50=0.11uM |
---|
Interaction Features: | 5 |
---|
|
+ | 83 | 3IKA | Epidermal growth factor receptor EGFR | ATP domain | 7.95 |
---|
Additional Details |
---|
Target Short Name: | EGFR |
---|
Cystal Resolution: | 2.9 Å |
---|
Reference Affinity: | IC50=14nM |
---|
Interaction Features: | 3 |
---|
|
+ | 84 | 5OQ6 | Serine/threonine-Transferase CHK1 | ATP domain | 7.95 |
---|
Additional Details |
---|
Target Short Name: | CHK1 |
---|
Cystal Resolution: | 1.95 Å |
---|
Reference Affinity: | Ki=0.0277uM |
---|
Interaction Features: | 5 |
---|
|
+ | 85 | 5N9L | Casein kinase ii subunit alpha | ATP domain | 7.94 |
---|
Additional Details |
---|
Target Short Name: | CK2alpha |
---|
Cystal Resolution: | 1.79 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 9 |
---|
|
+ | 86 | 2VX0 | Ephrin type-B receptor 4 EPHB4 | ATP domain | 7.93 |
---|
Additional Details |
---|
Target Short Name: | EPHB4 |
---|
Cystal Resolution: | 2.1 Å |
---|
Reference Affinity: | IC50=0.58uM |
---|
Interaction Features: | 5 |
---|
|
+ | 87 | 3QQU | Insulin-like growth factor 1 receptor precursor IGF1R | ATP domain | 7.93 |
---|
Additional Details |
---|
Target Short Name: | IGF1R |
---|
Cystal Resolution: | 2.9 Å |
---|
Reference Affinity: | IC50=2.4nM |
---|
Interaction Features: | 5 |
---|
|
+ | 88 | 2CDZ | Serine/threonine-protein kinase pak 4 | ATP domain | 7.93 |
---|
Additional Details |
---|
Target Short Name: | PAK4 |
---|
Cystal Resolution: | 2.30 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 5 |
---|
|
+ | 89 | 4J3I | Bromodomain-containing protein 4 | BRD domain | 7.90 |
---|
Additional Details |
---|
Target Short Name: | BRD4 |
---|
Cystal Resolution: | 1.24 Å |
---|
Reference Affinity: | IC50=1.8uM |
---|
Interaction Features: | 3 |
---|
|
+ | 90 | 3LFC | Mitogen-activated protein kinase 14 MAPK14 | ATP domain/Hydrophobic pocket | 7.90 |
---|
Additional Details |
---|
Target Short Name: | MAPK14 |
---|
Cystal Resolution: | 2.8 Å |
---|
Reference Affinity: | Kd=287nM |
---|
Interaction Features: | 7 |
---|
|
+ | 91 | 2R3P | Cyclin dependent kinase 2 CDK2 | ATP domain | 7.90 |
---|
Additional Details |
---|
Target Short Name: | CDK2 |
---|
Cystal Resolution: | 1.66 Å |
---|
Reference Affinity: | IC50=900nM |
---|
Interaction Features: | 5 |
---|
|
+ | 92 | 1E98 | Thymidylate kinase | ATP domain | 7.90 |
---|
Additional Details |
---|
Target Short Name: | DTYMK |
---|
Cystal Resolution: | 1.9 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 4 |
---|
|
+ | 93 | 5XDK | Epidermal growth factor receptor EGFR | ATP domain | 7.90 |
---|
Additional Details |
---|
Target Short Name: | EGFR |
---|
Cystal Resolution: | 2.346~ Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 4 |
---|
|
+ | 94 | 4BCF | Cyclin-dependent kinase 9 CDK9 | ATP domain | 7.90 |
---|
Additional Details |
---|
Target Short Name: | CDK9 |
---|
Cystal Resolution: | 3.01 Å |
---|
Reference Affinity: | Ki=7nM |
---|
Interaction Features: | 6 |
---|
|
+ | 95 | 3PRZ | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform | ATP domain | 7.90 |
---|
Additional Details |
---|
Target Short Name: | PIK3CG |
---|
Cystal Resolution: | 2.6 Å |
---|
Reference Affinity: | Ki=26nM |
---|
Interaction Features: | 6 |
---|
|
+ | 96 | 2VWZ | Ephrin type-B receptor 4 EPHB4 | ATP domain | 7.88 |
---|
Additional Details |
---|
Target Short Name: | EPHB4 |
---|
Cystal Resolution: | 1.65 Å |
---|
Reference Affinity: | IC50=0.794uM |
---|
Interaction Features: | 7 |
---|
|
+ | 97 | 2BDF | Proto-oncogene tyrosine-protein kinase Src | ATP domain | 7.88 |
---|
Additional Details |
---|
Target Short Name: | SRC |
---|
Cystal Resolution: | 2.1 Å |
---|
Reference Affinity: | IC50=0.067uM |
---|
Interaction Features: | 4 |
---|
|
+ | 98 | 3O51 | Aurora A kinase AurA | ATP domain/Hydrophobic pocket | 7.88 |
---|
Additional Details |
---|
Target Short Name: | AurA |
---|
Cystal Resolution: | 3.2 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 6 |
---|
|
+ | 99 | 4YJO | Tyrosine-protein kinase SYK | ATP domain | 7.88 |
---|
Additional Details |
---|
Target Short Name: | SYK |
---|
Cystal Resolution: | 1.6 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 7 |
---|
|
+ | 100 | 5XY1 | Tyrosine-protein kinase LYN | ATP domain | 7.88 |
---|
Additional Details |
---|
Target Short Name: | LYN |
---|
Cystal Resolution: | 2.7 Å |
---|
Reference Affinity: | ~ |
---|
Interaction Features: | 3 |
---|
|